RO-9187,HCV病毒复制抑制剂

RO-9187 (订货以英文为准)

编号:R127469
CAS号:876708-03-1
分子式:C9H12N6O5
分子量:284.23
货号 品牌 包装 目录价 您的价格 库存 数量 购买
R127469-5mg 阿拉丁 5mg ¥3353.90
R127469-50mg 阿拉丁 50mg ¥13938.90
R127469-10mg 阿拉丁 10mg ¥4389.90
产品名称 RO-9187
中文名称 RO-9187,HCV病毒复制抑制剂
CAS号 876708-03-1
分子式(M.F.) C9H12N6O5
分子量(M.W.) 284.23
储存条件 -20°C储存
溶解性DMSO
存贮条件储存温度-20°C
生化机理RO-9187 is a potent inhibitor of HCV virus replication in the replicon system (IC(50) = 171 +/- 12 nM; CC(50) >1 mM). Pharmacokinetic studies with RO-9187 in rats and dogs showed that plasma concentrations exceeding HCV replicon IC(50) values 8-150-fold could be achieved by low dose (10 mg/kg) oral administration.
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