溶解性 | Soluble in DMSO (17 mg/ml at 25 °C), water (<1 mg/ml at 25 °C), ethanol (<1 mg/ml at 25 °C), and 30% PEG400/0.5% Tween80/5% propylene glycol (30 mg/ml at 25 °C). |
存贮条件 | 储存温度-20°C |
应用 | A multi-targeted inhibitor. |
产品介绍 | Pazopanib HCl (GW786034 HCl)是一种新型的针对VEGFR-1, VEGFR-2, VEGFR-3, PDGFR, FGFR, c-Kit和c-fms等多个靶点的抑制剂,IC50分别是10 nM, 30 nM, 47 nM, 84 nM, 74 nM, 140 nM和146 nM。 |
备注 | Pazopanib (GW786034) is a novel multi-target inhibitor of VEGFR1, VEGFR2, VEGFR3, PDGFR, FGFR, c-Kit and c-Fms with IC50 of 10 nM, 30 nM, 47 nM, 84 nM, 74 nM, 140 nM and 146 nM, respectively.Phase 2 |
生化机理 | Pazopanib Hydrochloride (GW786034, Votrient, Armala) is a novel, multitargeted inhibitor of VEGFR-1, VEGFR-2, VEGFR-3, PDGFR, FGFR, c-Kit and c-fms with IC50 values of 10 nM, 30 nM, 47 nM, 84 nM, 74 nM, 140 nM and 146 nM, respectively. |
别名 | GW786034;盐酸帕唑帕尼;GW786034; Votrient; Armala; GW 786034; GW-786034;Pazopanib hydrochloride |
盐酸帕唑帕尼 (GW786034 HCl)
Pazopanib HCl (GW786034 HCl) (订货以英文为准)
编号:P129722
CAS号:635702-64-6
分子式:C21H24CLN7O2S
分子量:473.98
产品名称 | Pazopanib HCl (GW786034 HCl) |
中文名称 | 盐酸帕唑帕尼 (GW786034 HCl) |
CAS号 | 635702-64-6 |
分子式(M.F.) | C21H24CLN7O2S |
分子量(M.W.) | 473.98 |
储存条件 | -20°C储存 |
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