| 沸点 | 605.93 °C at 760 mmHg |
| 折光率 | 1.65 |
| 溶解性 | Soluble in DMSO, DMF, ethanol, water (0.2 mg/ml) at 25 °C, and 1:4 DMF:PBS(pH 7.2) (0.2 mg/ml). |
| 存贮条件 | 储存温度2-8℃ |
| 密度 | 1.5000 |
| 应用 | A selective CB2 receptor antagonist that binds to CB1 and CB2 receptors |
| 产品介绍 | AM630是CB2拮抗剂，Ki为31.2 nM，比对CB1受体的抑制性高150倍以上。 |
| 生化机理 | AM630 is a selectivity CB2 antagonist with Ki of 31.2 nM; > 150 fold selectivity over CB1 receptor.AM630 is a selective CB2 receptor antagonist that binds to CB1 and CB2 receptors with Ki values of 5.2 uM and 31.2 nM, respectively. AM630 has been shown to display 165-fold selectivity over CB1 receptors and behave as a weak partial/inverse agonist at CB1 receptors. AM630 acts as a cannabinoid receptor antagonist in mouse brain, vas deferens and guinea pig brain, but acts as an agonist in guinea pig leum. AM630 acts as an inverse agonist on cloned human CB1 receptors. |
| 别名 | AM 630;AM-630; [6-碘-2-甲基-1-[2-(4-吗啉基)乙基]-1H-吲哚-3-基](4-甲氧基苯基)甲酮;AM 630;AM-630; 6-Iodo-2-methyl-1-[2-(4-morpholinyl)ethyl]-1H-indol-3-yl](4-methoxyphenyl)methanone; Iodopravadoline |
AM630,CB2 大麻素拮抗剂/反向激动剂
AM630 （订货以英文为准）
编号：A124994
CAS号：164178-33-0
分子式：C23H25IN2O3
分子量：504.36
| 产品名称 | AM630 |
| 中文名称 | AM630,CB2 大麻素拮抗剂/反向激动剂 |
| CAS号 | 164178-33-0 |
| MDL编码 | MFCD01861183 |
| 分子式（M.F.） | C23H25IN2O3 |
| 分子量（M.W.） | 504.36 |
| 储存条件 | 2-8°C储存 |
| Reaxys-RN | 4552782 |
| 标识符号 | https://www.aladdin-e.com/images/ghs/ghs06.jpg |
| 信号词 | Danger |
| 危害声明 | H301 |
| 警示性声明 | P301 + P310 |
| WGK德国 | 3 |
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