PF-4981517,CYP3A4抑制剂

PF-4981517 (订货以英文为准)

编号:E129750
CAS号:1390637-82-7
分子式:C26H32N8
分子量:456.59
货号 品牌 包装 目录价 您的价格 库存 数量 购买
E129750-50mg 阿拉丁 50mg ¥7518.00
E129750-10mg 阿拉丁 10mg ¥1750.00
E129750-1mg 阿拉丁 1mg ¥399.90
E129750-5mg 阿拉丁 5mg ¥1499.90
E129750-100mg 阿拉丁 100mg ¥13698.00
产品名称 PF-4981517
中文名称 PF-4981517,CYP3A4抑制剂
CAS号 1390637-82-7
分子式(M.F.) C26H32N8
分子量(M.W.) 456.59
储存条件 -20°C储存
溶解性DMSO 91 mg/mL Water <1 mg/mL Ethanol <1 mg/mL
存贮条件储存温度-20°C
备注PF-4981517 is a potent and selective inhibitor of CYP3A4 (P450) with IC50 of 0.03 μM, exhibits >500-fold selectivity over CYP3A5 and CYP3A7.
别名PF-04981517;1H-Pyrazolo[3,4-d]pyrimidine, 1-methyl-3-[1-methyl-5-(4-methylphenyl)-1H-pyrazol-4-yl]-4-[(3S)-3-(1-piperidinyl)-1-pyrrolidinyl]-;PF-04981517;1H-Pyrazolo[3,4-d]pyrimidine, 1-methyl-3-[1-methyl-5-(4-methylphenyl)-1H-pyrazol-4-yl]-4-[(3S)-3-(1-piperidinyl)-1-pyrrolidinyl]-
标识符号https://www.aladdin-e.com/images/ghs/ghs07.jpg
信号词Warning
危害声明H302-H315-H319-H335
警示性声明P261-P305 + P351 + P338
个人防护设备dust mask type N95 (US), Eyeshields, Gloves
RTECSDM2953750
WGK德国3
搜索质检报告(COA)
搜索MSDS
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