溶解性 | DMSO 91 mg/mL Water <1 mg/mL Ethanol <1 mg/mL |
存贮条件 | 储存温度-20°C |
备注 | PF-4981517 is a potent and selective inhibitor of CYP3A4 (P450) with IC50 of 0.03 μM, exhibits >500-fold selectivity over CYP3A5 and CYP3A7. |
别名 | PF-04981517;1H-Pyrazolo[3,4-d]pyrimidine, 1-methyl-3-[1-methyl-5-(4-methylphenyl)-1H-pyrazol-4-yl]-4-[(3S)-3-(1-piperidinyl)-1-pyrrolidinyl]-;PF-04981517;1H-Pyrazolo[3,4-d]pyrimidine, 1-methyl-3-[1-methyl-5-(4-methylphenyl)-1H-pyrazol-4-yl]-4-[(3S)-3-(1-piperidinyl)-1-pyrrolidinyl]- |
PF-4981517,CYP3A4抑制剂
PF-4981517 (订货以英文为准)
编号:E129750
CAS号:1390637-82-7
分子式:C26H32N8
分子量:456.59
产品名称 | PF-4981517 |
中文名称 | PF-4981517,CYP3A4抑制剂 |
CAS号 | 1390637-82-7 |
分子式(M.F.) | C26H32N8 |
分子量(M.W.) | 456.59 |
储存条件 | -20°C储存 |
标识符号 | https://www.aladdin-e.com/images/ghs/ghs07.jpg |
信号词 | Warning |
危害声明 | H302-H315-H319-H335 |
警示性声明 | P261-P305 + P351 + P338 |
个人防护设备 | dust mask type N95 (US), Eyeshields, Gloves |
RTECS | DM2953750 |
WGK德国 | 3 |
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