Torcetrapib,胆固醇酯转移蛋白(CETP)抑制剂

Torcetrapib (订货以英文为准)

编号:E129832
CAS号:262352-17-0
分子式:C26H25N2O4F9
分子量:600.47
货号 品牌 包装 目录价 您的价格 库存 数量 购买
E129832-10mg 阿拉丁 10mg ¥969.90
E129832-50mg 阿拉丁 50mg ¥3193.90
E129832-5mg 阿拉丁 5mg ¥710.90
产品名称 Torcetrapib
中文名称 Torcetrapib,胆固醇酯转移蛋白(CETP)抑制剂
CAS号 262352-17-0
分子式(M.F.) C26H25N2O4F9
分子量(M.W.) 600.47
储存条件 2-8°C储存
溶解性Soluble in chloroform, methanol, ethanol (~10 mg/ml), DMSO (120 mg/ml at 25 °C), DMF (~20 mg/ml), and water (<1 mg/ml at 25 °C).
存贮条件储存温度2-8℃
应用A CETP inhibitor.
产品介绍Torcetrapib是一种CETP抑制剂,IC50为37 nM,提高血浆中HDL-C,降低nonHDL-C。Phase 3。
合法信息Sold for only research purposes
备注Torcetrapib is a CETP inhibitor with IC50 of 37 nM, elevates HDL-C and reduces nonHDL-C in plasma. Phase 3.
生化机理Torcetrapib is a CETP (cholesteryl ester transfer protein) inhibitor that is an antilipemic and antiatherosclerotic.
别名托彻普; (2R,4S)-4-[(3,5-双三氟甲基苄基)甲氧基甲酰氨基]-2-乙基-6-三氟甲基-3,4-二氢-2H-喹啉-1-羧酸乙酯;CP-529,414;CP-529414;(2R,4S)-4-((3,5-Bis-trifluoromethylbenzyl)methoxycarbonylamino)-2-ethyl-6-trifluoromethyl-3,4-dihydro-2H-quinoline-1-carboxylic acid ethyl ester
搜索质检报告(COA)
搜索MSDS
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