Nepicastat,抑制剂

Nepicastat (订货以英文为准)

编号:N125368
CAS号:173997-05-2
分子式:C14H15F2N3S
分子量:295.35
货号 品牌 包装 目录价 您的价格 库存 数量 购买
N125368-50mg 阿拉丁 50mg ¥11064.90
N125368-5mg 阿拉丁 5mg ¥1999.90
N125368-10mg 阿拉丁 10mg ¥3767.90
产品名称 Nepicastat
中文名称 Nepicastat,抑制剂
CAS号 173997-05-2
分子式(M.F.) C14H15F2N3S
分子量(M.W.) 295.35
储存条件 -20°C储存
溶解性DMSO
存贮条件储存温度-20°C
生化机理Nepicastat (SYN117; RS-25560-197) is a dopamine beta-hydroxylase inhibitor with IC50 of 8.5 ± 0.8 and 9.0 ± 0.8 nM for bovine and human, respectively. Dopamine beta-hydroxylase is an enzyme that catalyzes the conversion of dopamine to norepinephrine. Nepicastat (SYN117; RS-25560-197) has been studied as a possible treatment for congestive heart failure, and appears to be well tolerated as such.
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