BMS-536924,双重IR / IGF1R抑制剂

BMS-536924 (订货以英文为准)

编号:B126005
CAS号:468740-43-4
分子式:C25H26N5O3CL
分子量:479.96
货号 品牌 包装 目录价 您的价格 库存 数量 购买
B126005-1mg 阿拉丁 1mg ¥119.90
B126005-100mg 阿拉丁 100mg ¥2210.90
B126005-25mg 阿拉丁 25mg ¥695.90
B126005-5mg 阿拉丁 5mg ¥390.90
产品名称 BMS-536924
中文名称 BMS-536924,双重IR / IGF1R抑制剂
CAS号 468740-43-4
分子式(M.F.) C25H26N5O3CL
分子量(M.W.) 479.96
储存条件 -20°C储存;充氩
溶解性DMSO 96 mg/mL Water <1 mg/mL Ethanol <1 mg/mL
存贮条件储存温度-20°C
备注BMS-536924 is an ATP-competitive IGF-1R/IR inhibitor with IC50 of 100 nM/73 nM, modest activity for Mek, Fak, and Lck with very little activity for Akt1, MAPK1/2.
生化机理BMS-536924 is a small molecule ATP-competitive IGF-IR kinase inhibitor with with an IC50 of 80 nM.
搜索质检报告(COA)
搜索MSDS
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