氯卡色林盐酸盐

Lorcaserin HCl (订货以英文为准)

编号:L129791
CAS号:846589-98-8
分子式:C11H14CLN.HCL
分子量:232.15
货号 品牌 包装 目录价 您的价格 库存 数量 购买
L129791-50mg 阿拉丁 50mg ¥102.90
L129791-250mg 阿拉丁 250mg ¥218.90
L129791-5g 阿拉丁 5g ¥2179.90
L129791-1g 阿拉丁 1g ¥529.90
产品名称 Lorcaserin HCl
中文名称 氯卡色林盐酸盐
CAS号 846589-98-8
分子式(M.F.) C11H14CLN.HCL
分子量(M.W.) 232.15
存贮条件储存温度-20°C
产品介绍Lorcaserin HCl是一种选择性的人源5-HT2C受体完全激动剂,Ki值为15 nM
生化机理BELVIQ (lorcaserin hydrochloride) is a serotonin 2C receptor?agonist?for oral administration used for chronic weight management. Lorcaserin is a highly selective 5-HT2C receptor agonist developed for the treatment of obesity. In rats, lorcaserin led to dose-dependent wt. loss. Lorcaserin proved safe and well tolerated in healthy volunteers and obese patients. In a phase II clin. study, patients administered 20 mg/day lorcaserin achieved an av. wt. loss of 3.6 kg (7.9 lbs), which was significantly greater than the av. wt. loss of 0.3 kg (0.7 lbs) in the placebo group. A phase III clin. trial is ongoing to evaluate the long-term safety and efficacy of lorcaserin in patients with obesity.
别名绿卡色林盐酸盐; (R)-8-氯-1-甲基-2,3,4,5-四氢-1H-3-苯并氮杂卓盐酸盐;(R)-8-Chloro-1-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine hydrochloride
WGK德国3
搜索质检报告(COA)
搜索MSDS
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