溶解性 | 25°C: DMSO |
存贮条件 | 储存温度-20°C |
产品介绍 | AZD-3463是ALK/IGF1R抑制剂。 |
备注 | AZD3463 is a novel orally bioavailable ALK inhibitor with Ki of 0.75 nM, which also inhibits IGF1R with equivalent potency. |
生化机理 | AZD-3463 is an ALK/IGF1R inhibitor which overcomes multiple mechanisms of acquired resistance to crizotinib. |
别名 | ZD3463;AZD 3463; N-(4-(4-氨基-1-哌啶基)-2-甲氧基苯基)-5-氯-4-(1H-吲哚-3-基)-2-嘧啶胺;;AZD3463;AZD 3463;ALK/IGF1R inhibitor;N-(4-(4-amino-1-piperidinyl)-2-methoxyphenyl)-5-chloro-4-(1h-indol-3-yl)-2-pyrimidinamine; |
N-[4-(4-氨基-1-哌啶基)-2-甲氧基苯基]-5-氯-4-(1H-吲哚-3-基)-2-嘧啶胺
AZD3463 (订货以英文为准)
编号:A125664
CAS号:1356962-20-3
分子式:C24H25CLN6O
分子量:448.95
产品名称 | AZD3463 |
中文名称 | N-[4-(4-氨基-1-哌啶基)-2-甲氧基苯基]-5-氯-4-(1H-吲哚-3-基)-2-嘧啶胺 |
CAS号 | 1356962-20-3 |
分子式(M.F.) | C24H25CLN6O |
分子量(M.W.) | 448.95 |
储存条件 | -20°C储存 |
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